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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50000796
(4-cyclopropylmethyl-10-hydroxy-14-(4-methylene-5-o...)
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Affinity Data
IC50: 2.80nM
Assay Description:
inhibition of 1.0 nM [3H]- DAGO binding to guinea pig brain membrane opioid receptor mu
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Homo sapiens (Human))
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50000796
(4-cyclopropylmethyl-10-hydroxy-14-(4-methylene-5-o...)
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Affinity Data
IC50: 7.70nM
Assay Description:
Inhibition of [3H]DPDPE binding to guinea pig brain membrane Opioid receptor delta 1 at 1.0 nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type/Kappa-type/Mu-type opioid receptor
(Homo sapiens (Human))
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50000796
(4-cyclopropylmethyl-10-hydroxy-14-(4-methylene-5-o...)
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Affinity Data
IC50: 14nM
Assay Description:
Inhibition of 0.5 nM [3H]bremazocine binding to guinea pig brain membrane opioid receptors
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
DrugBank
antibodypedia
antibodypedia
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Washington
Curated by
ChEMBL
Ligand
BDBM50000796
(4-cyclopropylmethyl-10-hydroxy-14-(4-methylene-5-o...)
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Affinity Data
IC50: 25nM
Assay Description:
Displacement of 0.5 nM [3H]bremazocine from guinea pig brain membrane opioid receptor kappa with 100 nM DAGO and 100 nM DPDPE
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI