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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50307793
(4-Acetamidophenyl 2-(4-(2-(trifluoromethyl)pyridin...)
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Affinity Data
Ki: 160nM
Assay Description:
Inhibition of FAAH-mediated [3H]AEA hydrolysis in rat brain homogenate by time-dependent studies
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Fatty-acid amide hydrolase 1 [30-579]
(Rattus norvegicus (rat))
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50307793
(4-Acetamidophenyl 2-(4-(2-(trifluoromethyl)pyridin...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 100nM
Assay Description:
Inhibition of FAAH-mediated [3H]AEA hydrolysis in rat brain homogenate by liquid scintillation spectroscopy
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Monoglyceride lipase
(Homo sapiens (Human))
University Of Cagliari
Curated by
ChEMBL
Ligand
BDBM50307793
(4-Acetamidophenyl 2-(4-(2-(trifluoromethyl)pyridin...)
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Copy InChI
Affinity Data
IC50: 1.90E+3nM
Assay Description:
Inhibition of human recombinant MGL
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI