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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
39
hits in this display
Target
Receptor tyrosine-protein kinase erbB-2
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 11nM
Assay Description:
Inhibition of human N-terminal DYKDDDD tagged HER2 cytoplasmic domain amino acid 676 to 1255 expressed in baculovirus after 5 mins by scintillation c...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 11nM
Assay Description:
Inhibition of human N-terminal DYKDDDD tagged EGFR cytoplasmic domain amino acid 669 to 1210 expressed in baculovirus after 5 mins by scintillation c...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Receptor tyrosine-protein kinase erbB-2
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
Copy SMILES
Copy InChI
Affinity Data
IC50: 11nM
Assay Description:
Inhibition of human N-terminal DYKDDDD tagged HER2 cytoplasmic domain amino acid 676 to 1255 expressed in baculovirus after 5 mins by scintillation c...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
UniProtKB/SwissProt
B.MOAD
DrugBank
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CHEMBL
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Article
PubMed
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Target
Epidermal growth factor receptor
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
Copy SMILES
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Affinity Data
IC50: 11nM
Assay Description:
Inhibition of human N-terminal DYKDDDD tagged EGFR cytoplasmic domain amino acid 669 to 1210 expressed in baculovirus after 5 mins by scintillation c...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Receptor tyrosine-protein kinase erbB-4
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 160nM
Assay Description:
Inhibition of HER4 cytoplasmic domain after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
UniProtKB/SwissProt
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Target
Aurora kinase B
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 500nM
Assay Description:
Inhibition of N-terminal His6-tagged Aurora B expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
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Target
Dual specificity mitogen-activated protein kinase kinase 1
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 980nM
Assay Description:
Inhibition of N-terminal GST-tagged MEK1 after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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Target
Tyrosine-protein kinase Lck
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 1.30E+3nM
Assay Description:
Inhibition of LCK after 5 mins
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase Lyn
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 3.30E+3nM
Assay Description:
Inhibition of LYN B after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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Target
Tyrosine-protein kinase Lyn
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 3.60E+3nM
Assay Description:
Inhibition of LYN A after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
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KEGG
UniProtKB/SwissProt
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Target
Hepatocyte growth factor receptor
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 3.90E+3nM
Assay Description:
Inhibition of c-Met after 5 mins
More data for this Ligand-Target Pair
Target Info
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Target
Tyrosine-protein kinase CSK
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: 5.10E+3nM
Assay Description:
Inhibition of CSK after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Glycogen synthase kinase-3 beta
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged GSK3beta expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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Target
Fibroblast growth factor receptor 1
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of FGFR1 after 5 min
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
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Target
Fibroblast growth factor receptor 3
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of FGFR3 after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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Article
PubMed
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Target
Proto-oncogene tyrosine-protein kinase Src
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of Src after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
Details
Article
PubMed
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Target
Mitogen-activated protein kinase kinase kinase 1
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of C-terminal FLAG-tagged MEKK expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Dual specificity protein kinase TTK
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged TTK expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Insulin-like growth factor 1 receptor
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of IGF-1R after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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Article
PubMed
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Target
Inhibitor of nuclear factor kappa-B kinase subunit beta
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of C-terminal FLAG-tagged IKKbeta expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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PC sid
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In Depth
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Article
PubMed
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Target
Mitogen-activated protein kinase 3
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged ERK1 expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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Target
Focal adhesion kinase 1
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of full length N-terminal FLAG-tagged FAK expressed in baculovirus after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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GoogleScholar
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CHEMBL
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PC sid
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Article
PubMed
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Target
Mitogen-activated protein kinase kinase kinase 5
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged ASK1 expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
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Article
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Target
Mitogen-activated protein kinase 14
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged p38alpha expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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PC sid
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In Depth
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Article
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Target
Insulin receptor
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of INSR after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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CHEMBL
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Article
PubMed
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Target
Angiopoietin-1 receptor
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of TIE2 after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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Article
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Target
Serine/threonine-protein kinase PLK1
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged PLK1 expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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Article
PubMed
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Target
Dual specificity mitogen-activated protein kinase kinase 5
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged MEK5 expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
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Target
Protein kinase C theta type
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged PKCtheta expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
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GoogleScholar
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CHEMBL
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Article
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Target
Mitogen-activated protein kinase 8
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged JNK1 expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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GoogleScholar
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CHEMBL
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Target
Mast/stem cell growth factor receptor Kit
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of c-kit after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
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CHEMBL
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Target
Tyrosine-protein kinase ZAP-70
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of ZAP70 after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
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GoogleScholar
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PC sid
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Article
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Target
Serine/threonine-protein kinase B-raf
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged B-raf expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
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CHEMBL
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Article
PubMed
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Target
Mitogen-activated protein kinase kinase kinase 7
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged TAK1 expressed in baculovirus after 5 mins by scintillation counter
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
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antibodypedia
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Target
Vascular endothelial growth factor receptor 1
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of VEGFR1 after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
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In Depth
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Article
PubMed
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Target
Vascular endothelial growth factor receptor 2
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of N-terminal FLAG-tagged VEGFR2 cytoplasmic domain expressed in baculovirus after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Platelet-derived growth factor receptor beta
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
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Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PDGFRbeta after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Platelet-derived growth factor receptor alpha
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of PDGFRalpha after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Cytoplasmic tyrosine-protein kinase BMX
(Homo sapiens (Human))
Takeda Pharmaceutical
Curated by
ChEMBL
Ligand
BDBM50391643
(CHEMBL2148052 | CHEMBL2148053)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.00E+4nM
Assay Description:
Inhibition of full length N-terminal FLAG-tagged BMX expressed in baculovirus after 5 mins
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI