Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBeta-3 adrenergic receptor(Canis familiaris)
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50264709((R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamin...)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at dog cloned adrenergic beta3 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-1 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50264709((R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamin...)
Affinity DataEC50:  620nMAssay Description:Agonist activity at human cloned adrenergic beta1 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-3 adrenergic receptor(Homo sapiens (Human))
Astellas Pharma

Curated by ChEMBL
LigandPNGBDBM50264709((R)-5-(3-(2-(2-(3-chlorophenyl)-2-hydroxyethylamin...)
Affinity DataEC50:  4.60nMAssay Description:Agonist activity at human cloned adrenergic beta3 receptor expressed in CHO cells assessed as cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed