Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158761(1-tert-Butyl-3-(2-furan-2-yl-8-phenethyl-8H-pyrazo...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity for human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158761(1-tert-Butyl-3-(2-furan-2-yl-8-phenethyl-8H-pyrazo...)
Affinity DataKi:  4.90nMAssay Description:Binding affinity to human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158761(1-tert-Butyl-3-(2-furan-2-yl-8-phenethyl-8H-pyrazo...)
Affinity DataKi:  4.90nMAssay Description:Antagonist activity at human adenosine A3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A3(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50158761(1-tert-Butyl-3-(2-furan-2-yl-8-phenethyl-8H-pyrazo...)
Affinity DataKi:  4.90E+3nMAssay Description:Displacement of [3H]MRE3008-F20 from human adenosine A3 receptor expressed in CHO cells after 120 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed