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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNeuromedin-K receptor(GUINEA PIG)
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  22nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
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TargetNeuromedin-K receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  22nMAssay Description:Binding affinity for NK3 receptor binding sites in guinea pig cortical membranes by using [125I][MePhe7]-NKB as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-K receptor(HAMSTER)
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  6.16E+3nMAssay Description:Binding affinity for NK2 receptor binding sites in membranes prepared from hamster urinary bladder by using [125I]NKA as radioligandMore data for this Ligand-Target Pair
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TargetSubstance-P receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50282782(CHEMBL297327 | {(S)-1-[(R)-1-(8-Hydroxy-octylcarba...)
Affinity DataIC50:  1.00E+4nMAssay Description:Binding affinity for NK1 receptor binding sites in human lymphoma IM9 cells by using [125I]-Bolton-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails Article