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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetAcetyl-CoA carboxylase 2(Homo sapiens (Human))
Astrazeneca Research And Development

Curated by ChEMBL
LigandPNGBDBM50350750(CHEMBL1818300)
Affinity DataIC50:  99nMAssay Description:Inhibition of human recombinant his-tagged ACC2 expressed in baculovirus/Sf9 cell assessed as inorganic phosphate formation preincubated for 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase(Rattus norvegicus (Rat))
Astrazeneca Research And Development

Curated by ChEMBL
LigandPNGBDBM50350750(CHEMBL1818300)
Affinity DataIC50:  150nMAssay Description:Inhibition of ACC2 in obese Zucker rat assessed as reduction in hepatic malonyl-coA level preincubated for 15 mins measured after 1.5 hrs using Malac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase 1(Rattus norvegicus (Rat))
Astrazeneca Research And Development

Curated by ChEMBL
LigandPNGBDBM50350750(CHEMBL1818300)
Affinity DataIC50:  250nMAssay Description:Inhibition of obese Zucker rat ACC1 assessed as reduction in hepatic malonyl-coA level preincubated for 15 mins measured after 1.5 hrs using Malachit...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetyl-CoA carboxylase 1(Homo sapiens (Human))
Astrazeneca Research And Development

Curated by ChEMBL
LigandPNGBDBM50350750(CHEMBL1818300)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of human recombinant his-tagged ACC1 expressed in baculovirus/Sf9 cell assessed as inorganic phosphate formation preincubated for 15 mins ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Astrazeneca Research And Development

Curated by ChEMBL
LigandPNGBDBM50350750(CHEMBL1818300)
Affinity DataIC50: >3.30E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed