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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Glucocorticoid receptor
(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50201096
(1-[2-hydroxy-4-(2-hydroxyphenyl)-4-methyl-2-(trifl...)
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Affinity Data
IC50: 6nM
Assay Description:
Inhibition of tetramethylrhodamine labeled dexamethosone binding to GR by FP assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mineralocorticoid receptor
(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50201096
(1-[2-hydroxy-4-(2-hydroxyphenyl)-4-methyl-2-(trifl...)
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Affinity Data
IC50: 450nM
Assay Description:
Inhibition of tetramethylrhodamine labeled dexamethosone binding to MR by FP assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Progesterone receptor
(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50201096
(1-[2-hydroxy-4-(2-hydroxyphenyl)-4-methyl-2-(trifl...)
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Copy InChI
Affinity Data
IC50: 555nM
Assay Description:
Inhibition of tetramethylrhodamine labeled RU486 binding to PR by FP assay
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI