Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetMetabotropic glutamate receptor 1(RAT)
Pfizer

Curated by ChEMBL

LigandBDBM50197262(CHEMBL246025 | N-(2-methyl-2-(pyridin-2-yl)propyl)...)Copy SMILESCopy InChI

Affinity DataKi:  40nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as increase in calcium internalisation by FLIPR assayMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
GoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
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