Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 13 hits in this display
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
EC50: 250nMAssay Description:Agonist activity at human LXR-beta expressed in African green monkey CV1 cells measured after 18 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
EC50: 220nMAssay Description:Agonist activity at human LXR-alpha expressed in African green monkey CV1 cells measured after 18 to 20 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
EC50: 33nMAssay Description:Agonist activity at LXR-beta in human HeLa cells assessed as induction of ABCA1 by beta-galactosidase/luciferase reporter gene assayMore data for this Ligand-Target Pair
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
EC50: 630nMAssay Description:As used herein, reference to the activity of an LXR agonist at LXRα and LXRβ refer to the activity as measured using the ligand sensing ass...More data for this Ligand-Target Pair
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
EC50: 550nMAssay Description:As used herein, reference to the activity of an LXR agonist at LXRα and LXRβ refer to the activity as measured using the ligand sensing ass...More data for this Ligand-Target Pair
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)
BDBM50034775(CHEMBL3360975 | US10543183, Compound 38 | US109459...)