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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDelta-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  0.120nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]-DPDPE (6.3 nM) for Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
National Institute Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataKi:  1.02E+3nMAssay Description:Affinity of the compound was assessed using competitive binding assay labeled with [3H]- DAGO (1.28 nM) for Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
National Institute Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50:  1.44nMAssay Description:Functional biological activity for Opioid receptor delta 1 was determined in vitro, on mouse vas deferens (MVD).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
National Institute Of Environmental Health Sciences

Curated by ChEMBL
LigandPNGBDBM50059370((S)-3-((S)-2-{2-[(S)-2-Amino-3-(4-hydroxy-phenyl)-...)
Affinity DataIC50: >10nMAssay Description:Functional biological activity for mu opioid receptor was determined in vitro , on guinea pig ileum (GPI).More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed