Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataKi:  0.241nMAssay Description:Displacement of [3H]deltorphin 2 from delta opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataKi:  154nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor in Sprague-Dawley rat brain P2 synaptosomal membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(MOUSE)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataIC50:  0.400nMAssay Description:Agonist activity at delta opioid receptor in mouse vas deferenceMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Cagliari

Curated by ChEMBL
LigandPNGBDBM50324024((2S,5S,8R,11S,14S)-2-amino-14-((S)-1-((S)-1-(2-ami...)
Affinity DataIC50:  3.56E+3nMAssay Description:Agonist activity at mu opioid receptor in Hartley guinea pig small intestineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed