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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNeprilysin(Rattus norvegicus (Rat))
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50048319((S)-3-Biphenyl-4-yl-2-{[1-((S)-2-mercapto-3-methyl...)
Affinity DataIC50:  16nMAssay Description:Evaluation of in vitro inhibitory activity against Neutral endopeptidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50048319((S)-3-Biphenyl-4-yl-2-{[1-((S)-2-mercapto-3-methyl...)
Affinity DataIC50:  77nMAssay Description:In vitro inhibition of human Endothelin converting Enzyme-1 activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEndothelin-converting enzyme 1(Homo sapiens (Human))
Novartis Institute For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50048319((S)-3-Biphenyl-4-yl-2-{[1-((S)-2-mercapto-3-methyl...)
Affinity DataIC50:  77nMAssay Description:In vitro inhibition of Endothelin-converting enzyme 1.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
Ciba-Geigy

Curated by ChEMBL
LigandPNGBDBM50048319((S)-3-Biphenyl-4-yl-2-{[1-((S)-2-mercapto-3-methyl...)
Affinity DataIC50:  139nMAssay Description:Evaluation of in vitro inhibitory activity against Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed