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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
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Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
Vitae Pharmaceuticals
US Patent
Ligand
BDBM168079
(US9073931, E27a | US9073931, E7a)
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Affinity Data
Ki: 2nM ΔG°: -49.7kJ/mole
T: 2°C
Assay Description:
Compounds of the invention were assessed in a competition binding assay where different concentrations of compounds were incubated with the LXR ligan...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
Vitae Pharmaceuticals
US Patent
Ligand
BDBM168079
(US9073931, E27a | US9073931, E7a)
Copy SMILES
Copy InChI
Affinity Data
Ki: 14nM ΔG°: -44.8kJ/mole
T: 2°C
Assay Description:
Compounds of the invention were assessed in a competition binding assay where different concentrations of compounds were incubated with the LXR ligan...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
Vitae Pharmaceuticals
US Patent
Ligand
BDBM168079
(US9073931, E27a | US9073931, E7a)
Copy SMILES
Copy InChI
Affinity Data
Ki: 23nM ΔG°: -43.6kJ/mole
T: 2°C
Assay Description:
Compounds of the invention were assessed in a competition binding assay where different concentrations of compounds were incubated with the LXR ligan...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
Vitae Pharmaceuticals
US Patent
Ligand
BDBM168079
(US9073931, E27a | US9073931, E7a)
Copy SMILES
Copy InChI
Affinity Data
Ki: 253nM ΔG°: -37.7kJ/mole
T: 2°C
Assay Description:
Compounds of the invention were assessed in a competition binding assay where different concentrations of compounds were incubated with the LXR ligan...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
Similars
In Depth
Details
US Patent
Copy BDB DOI