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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50035944(2-(3-Benzenesulfonylamino-2-oxo-6-phenyl-2H-pyridi...)
Affinity DataKi:  6nMAssay Description:Binding affinity against human leukocyte elastase (HLE) enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Zeneca Pharmaceuticals Group

Curated by ChEMBL
LigandPNGBDBM50035944(2-(3-Benzenesulfonylamino-2-oxo-6-phenyl-2H-pyridi...)
Affinity DataKi:  6nMAssay Description:In vitro inhibition constant (Ki) against human leukocyte elastase (HLE-catalyzed hydrolysis of MeO-Suc-Ala-Ala-Pro-Ala-pNA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed