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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Mitogen-activated protein kinase kinase kinase 12
(Homo sapiens (Human))
The University Of Texas System
US Patent
Ligand
BDBM289427
((R)-1-(4-(6-amino-5-(trifluoromethoxy)pyridin-3-yl...)
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Affinity Data
Kd: 45nM
Assay Description:
The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
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Target
Mitogen-activated protein kinase kinase kinase 12
(Homo sapiens (Human))
The University Of Texas System
US Patent
Ligand
BDBM590004
((S)-1-(4-(6-amino-5- (trifluoromethoxy)pyridin-3-y...)
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Affinity Data
Kd: 0.290nM
Assay Description:
A fusion protein of full length of human DLK (amino acids 1-859) and the DNA binding domain of NFkB was expressed in transiently transfected HEK293 c...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
PDB
3D Structure (crystal)
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Target
Mitogen-activated protein kinase kinase kinase 12
(Homo sapiens (Human))
The University Of Texas System
US Patent
Ligand
BDBM289495
(1-(4-(6-amino-5-(tri- fluoromethyl)pyridin-3- yl)-...)
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Affinity Data
Kd: 0.110nM
Assay Description:
The DLK dissociation constants (Kd) have been determined in the KINOMEscan KdELECT Service at DiscoveRx. A fusion protein of full length of human DLK...
More data for this Ligand-Target Pair
Target Info
PDB
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
PDB
In Depth
Details
US Patent
PDB
3D Structure (crystal)
Copy BDB DOI