Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 37 hits in this display
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
IC50: >2.00E+4nMAssay Description:Time dependent inhibition of CYP34A (unknown origin) using BFC as substrate incubated for 30 mins in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
IC50: >2.00E+4nMAssay Description:Time dependent inhibition of CYP34A (unknown origin) using BFC as substrate incubated for 5 mins in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
IC50: >2.00E+4nMAssay Description:Inhibition of CYP34A (unknown origin) using BFC as substrate incubated for 10 mins in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
IC50: >4.00E+4nMAssay Description:Time dependent inhibition of CYP34A (unknown origin) using TST as substrate incubated for up to 30 mins in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
IC50: >4.00E+4nMAssay Description:Time dependent inhibition of CYP34A (unknown origin) using MDZ as substrate incubated for up to 30 mins in presence of NADPH by LC-MS/MS analysisMore data for this Ligand-Target Pair
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)
BDBM311268((S)-1-((2′,4-bis(difluoromethyl)-[2,4′...)