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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM311368
((S)-1-((5-(7-chloroquinolin-4-yl)-3-methylpyridin-...)
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Copy InChI
Affinity Data
IC50: 0.740nM
Assay Description:
The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM311368
((S)-1-((5-(7-chloroquinolin-4-yl)-3-methylpyridin-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.740nM
Assay Description:
The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM311368
((S)-1-((5-(7-chloroquinolin-4-yl)-3-methylpyridin-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.740nM
Assay Description:
The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM311368
((S)-1-((5-(7-chloroquinolin-4-yl)-3-methylpyridin-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.740nM
Assay Description:
The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM311368
((S)-1-((5-(7-chloroquinolin-4-yl)-3-methylpyridin-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.740nM
Assay Description:
The assays were performed in U-bottom 384-well plates. The final assay volume was 30 Cl prepared from 15 μl additions of enzyme and substrates (...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI
Target
AP2-associated protein kinase 1
(Homo sapiens (Human))
Bristol-Myers Squibb
US Patent
Ligand
BDBM311368
((S)-1-((5-(7-chloroquinolin-4-yl)-3-methylpyridin-...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 0.740nM
Assay Description:
The assays were performed in U-bottom 384-well plates. The final assay volume was 30 μl prepared from 15 μl additions of enzyme and substra...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
PC cid
PC sid
In Depth
Details
US Patent
Copy BDB DOI