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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Mu-type opioid receptor
(Rattus norvegicus (rat))
University Of Paris
Curated by
ChEMBL
Ligand
BDBM50018714
(2-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
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Affinity Data
Ki: 116nM
Assay Description:
Inhibition of [3H]DAGO binding to mu 1 opioid receptor in rat brain membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Rattus norvegicus (rat))
University Of Paris
Curated by
ChEMBL
Ligand
BDBM50018714
(2-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
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Copy InChI
Affinity Data
Ki: 3.81E+3nM
Assay Description:
Inhibition of [3H]DSLET binding to delta 1 opioid receptors in rat brain membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Paris
Curated by
ChEMBL
Ligand
BDBM50018714
(2-[(2-{2-[2-Amino-3-(4-hydroxy-phenyl)-propionylam...)
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Copy InChI
Affinity Data
IC50: 379nM
Assay Description:
Inhibition of electrically evoked contraction of guinea pig ileum (myenteric plexus:longitudinal muscle preparation) by antagonist action at mu 1 opi...
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
KEGG
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI