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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Matrix metalloproteinase-9
(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by
ChEMBL
Ligand
BDBM50040579
((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
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Affinity Data
IC50: 15nM
Assay Description:
Activity against human gelatinase (MMP-9).
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Interstitial collagenase
(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by
ChEMBL
Ligand
BDBM50040579
((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
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Copy InChI
Affinity Data
IC50: 41nM
Assay Description:
Activity against human collagenase (MMP-1).
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Stromelysin-1
(Homo sapiens (Human))
Glaxo Inc. Research Institute
Curated by
ChEMBL
Ligand
BDBM50040579
((R)-4-(1,3-Dioxo-1,3-dihydro-benzo[f]isoindol-2-yl...)
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Copy InChI
Affinity Data
IC50: 1.49E+3nM
Assay Description:
Activity against human stromelysin (MMP-3).
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI