Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

Target72 kDa type IV collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285562((R)-2-[(S)-3-(3,5-Dimethyl-phenyl)-1-((S)-3-methyl...)
Affinity DataKi:  4.84E+3nMAssay Description:Inhibitory activity against human gelatinase-A (MMP-2)More data for this Ligand-Target Pair
In DepthDetails Article
TargetInterstitial collagenase(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285562((R)-2-[(S)-3-(3,5-Dimethyl-phenyl)-1-((S)-3-methyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against human collagenase (MMP-1)More data for this Ligand-Target Pair
In DepthDetails Article
TargetStromelysin-1(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50285562((R)-2-[(S)-3-(3,5-Dimethyl-phenyl)-1-((S)-3-methyl...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibitory activity against human stromelysin-3 (MMP-3)More data for this Ligand-Target Pair
In DepthDetails Article