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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Proteasome subunit beta type-5
(Homo sapiens (Human))
Gorlaeus Laboratories
Curated by
ChEMBL
Ligand
BDBM50307483
((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
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Affinity Data
IC50: 100nM
Assay Description:
Inhibition of 26S proteasome beta 5 using LLVY as substrate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-1
(Homo sapiens (Human))
Gorlaeus Laboratories
Curated by
ChEMBL
Ligand
BDBM50307483
((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
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Copy InChI
Affinity Data
IC50: >1.50E+4nM
Assay Description:
Inhibition of 26S proteasome beta 1 using nLPnLD as substrate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Proteasome subunit beta type-2
(Homo sapiens (Human))
Gorlaeus Laboratories
Curated by
ChEMBL
Ligand
BDBM50307483
((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
Copy SMILES
Copy InChI
Affinity Data
IC50: >1.50E+4nM
Assay Description:
Inhibition of 26S proteasome beta 2 using RLR as substrate
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI