Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetProteasome subunit beta type-5(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307483((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
Affinity DataIC50:  100nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307483((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307483((S)-2-azido-N-((S)-1-((S)-3-(3,5-bis(trifluorometh...)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed