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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 15 hits in this display   

TargetProteasome subunit beta type-5(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  1nMAssay Description:Inhibition of 26S proteasome beta 5 using LLVY as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta5 in human Raji cells incubated for 1 hr by BODIPY(TMR)-NC-005-VS probe b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  2.10nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta5 in human Raji cells incubated for 1 hr by BODIPY(TMR)-NC-005-VS probe b...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta5 in human Raji cells incubated for 1 hr by BODIPY(TMR)-NC-005-VS probe based co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Gorlaeus Laboratories

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  5.5nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta5 in human Raji cells incubated for 1 hr by BODIPY(TMR)-NC-005-VS probe based co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  13nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  13nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  66nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  67nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  120nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta1 in human Raji cells incubated for 1 hr by Cy5-NC-001 probe based competitive a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  123nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta1 in human Raji cells incubated for 1 hr by Cy5-NC-001 probe based competitive a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of 26S proteasome beta 2 using RLR as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: >1.50E+4nMAssay Description:Inhibition of 26S proteasome beta 1 using nLPnLD as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta1 in human Raji cells incubated for 1 hr by Cy5-NC-001 probe based compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Leiden Institute Of Chemistry

Curated by ChEMBL
LigandPNGBDBM50307481((S)-2-azido-N-((S)-1-((S)-1-((S)-4-methyl-1-((R)-2...)
Affinity DataIC50: <1.00E+5nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta1 in human Raji cells incubated for 1 hr by Cy5-NC-001 probe based compet...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed