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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
5
hits in this display
Target
Kappa-type opioid receptor
(Cavia porcellus (domestic guinea pig))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50040131
(CHEMBL409793 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-c((D-Cy...)
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Affinity Data
IC50: 0.116nM
Assay Description:
Inhibition of [3H]-U-69,593 binding to kappa opoid receptor of guinea pig brain homogenate
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50040131
(CHEMBL409793 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-c((D-Cy...)
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Affinity Data
IC50: 0.674nM
Assay Description:
Inhibition of [3H]-PL-17 binding to mu opioid receptor of guinea pig brain homogenate
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(GUINEA PIG)
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50040131
(CHEMBL409793 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-c((D-Cy...)
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Affinity Data
IC50: 4.5nM
Assay Description:
Inhibition of mu-selective antagonist binding to opioid receptor of guinea pig ileum
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Homo sapiens (Human))
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50040131
(CHEMBL409793 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-c((D-Cy...)
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Affinity Data
IC50: 6.5nM
Assay Description:
Inhibition of [3H]-DPDPE binding to delta opioid receptor of guinea pig brain homogenate
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(MOUSE)
University Of Arizona
Curated by
ChEMBL
Ligand
BDBM50040131
(CHEMBL409793 | Tyr-Gly-Gly-Phe-Leu-Arg-Arg-c((D-Cy...)
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Affinity Data
IC50: 25.3nM
Assay Description:
Inhibition of delta-selective antagonist binding to opioid receptor of mouse vas dferens
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI