Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetPlasminogen(Rattus norvegicus)
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013004(2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl...)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of plasminMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013004(2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl...)
Affinity DataIC50:  5.20E+3nMAssay Description:Evaluated for the inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKallikrein-1(Homo sapiens (Human))
University Of Arkansas

Curated by ChEMBL
LigandPNGBDBM50013004(2-Acetylamino-4-methyl-pentanoic acid [1-(1-formyl...)
Affinity DataIC50:  3.24E+4nMAssay Description:Inhibition of Kallikrein proteolytic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed