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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
3
hits in this display
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50220698
((R)-N-((S)-3-(4-chlorophenyl)-1-(4-(cyanomethyl)-4...)
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Affinity Data
IC50: 63nM
Assay Description:
Binding affinity to human MC4R
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 5
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50220698
((R)-N-((S)-3-(4-chlorophenyl)-1-(4-(cyanomethyl)-4...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 1.10E+3nM
Assay Description:
Antagonist activity at human MC5R assessed as stimulation of cAMP production
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Melanocortin receptor 4
(Homo sapiens (Human))
Merck
Curated by
ChEMBL
Ligand
BDBM50220698
((R)-N-((S)-3-(4-chlorophenyl)-1-(4-(cyanomethyl)-4...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 827nM
Assay Description:
Antagonist activity at human MC4R assessed as stimulation of cAMP production
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI