Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 6 hits in this display   

TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50153131(CHEMBL185415 | {1-[1-(4-Isopropyl-cyclohexyl)-pipe...)
Affinity DataKi:  25nMAssay Description:Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50153131(CHEMBL185415 | {1-[1-(4-Isopropyl-cyclohexyl)-pipe...)
Affinity DataKi:  33nMAssay Description:Inhibition of [3H]nociceptin binding to human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50153131(CHEMBL185415 | {1-[1-(4-Isopropyl-cyclohexyl)-pipe...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of [3H]U-69593 binding to human Opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50153131(CHEMBL185415 | {1-[1-(4-Isopropyl-cyclohexyl)-pipe...)
Affinity DataKi: >2.00E+3nMAssay Description:Inhibition of [3H]naltrindole binding to human Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50153131(CHEMBL185415 | {1-[1-(4-Isopropyl-cyclohexyl)-pipe...)
Affinity DataEC50:  227nMAssay Description:Agonist activity as stimulation of [35S]-GTP-gamma binding to human Opioid receptor like 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50153131(CHEMBL185415 | {1-[1-(4-Isopropyl-cyclohexyl)-pipe...)
Affinity DataEC50:  344nMAssay Description:Agonist activity as stimulation of [35S]-GTP-gamma binding to human Opioid receptor mu 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed