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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
6
hits in this display
Target
Nociceptin receptor
(Homo sapiens (Human))
Purdue Pharma
Curated by
ChEMBL
Ligand
BDBM50153127
(2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2...)
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Affinity Data
Ki: 3.90nM
Assay Description:
Inhibition of [3H]nociceptin binding to human Opioid receptor like 1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Mu-type opioid receptor
(Homo sapiens (Human))
Purdue Pharma
Curated by
ChEMBL
Ligand
BDBM50153127
(2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2...)
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Affinity Data
Ki: 92nM
Assay Description:
Inhibition of [3H]diprenorphine binding to human Opioid receptor mu 1
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Delta-type opioid receptor
(Homo sapiens (Human))
Purdue Pharma
Curated by
ChEMBL
Ligand
BDBM50153127
(2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2...)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of [3H]naltrindole binding to human Opioid receptor delta 1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
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Target
Kappa-type opioid receptor
(Homo sapiens (Human))
Purdue Pharma
Curated by
ChEMBL
Ligand
BDBM50153127
(2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2...)
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Affinity Data
Ki: >2.00E+3nM
Assay Description:
Inhibition of [3H]U-69593 binding to human Opioid receptor kappa 1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Mu-type opioid receptor
(Homo sapiens (Human))
Purdue Pharma
Curated by
ChEMBL
Ligand
BDBM50153127
(2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2...)
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Copy InChI
Affinity Data
EC50: 555nM
Assay Description:
Agonist activity as stimulation of [35S]-GTP-gamma binding to human Opioid receptor mu 1
More data for this Ligand-Target Pair
Target Info
PDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Nociceptin receptor
(Homo sapiens (Human))
Purdue Pharma
Curated by
ChEMBL
Ligand
BDBM50153127
(2-{1-[1-(4-Isopropyl-cyclohexyl)-piperidin-4-yl]-2...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 22nM
Assay Description:
Agonist activity as stimulation of [35S]-GTP-gamma binding to human Opioid receptor like 1
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI