Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

TargetNociceptin receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50132639(1-(4-Isopropyl-cyclohexyl)-4-(3-trifluoromethyl-ph...)
Affinity DataKi:  12nMAssay Description:Antagonistic activity against orphan FQ receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50132639(1-(4-Isopropyl-cyclohexyl)-4-(3-trifluoromethyl-ph...)
Affinity DataKi:  36nMAssay Description:Antagonistic activity against opioid receptor mu1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50132639(1-(4-Isopropyl-cyclohexyl)-4-(3-trifluoromethyl-ph...)
Affinity DataKi:  4.15E+3nMAssay Description:Antagonistic activity of the compound against opioid receptor kappa 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Purdue Pharma

Curated by ChEMBL
LigandPNGBDBM50132639(1-(4-Isopropyl-cyclohexyl)-4-(3-trifluoromethyl-ph...)
Affinity DataKi:  5.67E+3nMAssay Description:Antagonistic activity against Opioid receptor delta 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed