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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Metabotropic glutamate receptor 3
(Rattus norvegicus (Rat))
Sanford-Burnham Medical Research Institute
Curated by
ChEMBL
Ligand
BDBM50017248
(CHEMBL3287689 | US10099993, Compound 38)
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Affinity Data
EC50: >1.00E+4nM
Assay Description:
Positive allosteric modulation of rat mGluR3 receptor expressed in HEK293 cells assessed as potentiation of glutamate-induced thallium flux incubated...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
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In Depth
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Article
PubMed
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Target
Metabotropic glutamate receptor 3
(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
US Patent
Ligand
BDBM50017248
(CHEMBL3287689 | US10099993, Compound 38)
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Copy InChI
Affinity Data
EC50: >1.00E+4nM
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
US Patent
Ligand
BDBM50017248
(CHEMBL3287689 | US10099993, Compound 38)
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Copy InChI
Affinity Data
EC50: 454nM
pH: 7.3 T: 2°C
Assay Description:
Human Embryonic Kidney (HEK-293) cell lines co-expressing rat mGlu receptors 2, 3, 4, 6, 7 or 8 and G protein-coupled inwardly-rectifying potassium (...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
US Patent
Copy BDB DOI
Target
Metabotropic glutamate receptor 2
(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute
US Patent
Ligand
BDBM50017248
(CHEMBL3287689 | US10099993, Compound 38)
Copy SMILES
Copy InChI
Affinity Data
EC50: 454nM
Assay Description:
Positive allosteric modulation of rat mGluR2 receptor expressed in HEK293 cells assessed as potentiation of glutamate-induced thallium flux incubated...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI