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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM84742(CAS_106650-56-0 | NSC_5210 | sibutramine)
Affinity DataKi:  2.14E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Boots Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM84742(CAS_106650-56-0 | NSC_5210 | sibutramine)
Affinity DataKi:  3.13E+3nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2B(Homo sapiens (Human))
Vernalis Research

Curated by PDSP Ki Database
LigandPNGBDBM84742(CAS_106650-56-0 | NSC_5210 | sibutramine)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2C(Homo sapiens (Human))
Vernalis Research

Curated by PDSP Ki Database
LigandPNGBDBM84742(CAS_106650-56-0 | NSC_5210 | sibutramine)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Vernalis Research

Curated by PDSP Ki Database
LigandPNGBDBM84742(CAS_106650-56-0 | NSC_5210 | sibutramine)
Affinity DataKi: >1.00E+4nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed