Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 1 hits in this display   

TargetAndrogen receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

LigandBDBM18545(7-[(2-methylpropyl)amino]-4-(trifluoromethyl)-1,2-...)Copy SMILESCopy InChI

Affinity DataKi:  65nM ΔG°:  -42.7kJ/mole IC50:  74nMpH: 7.4 T: 2°CAssay Description:The compounds were evaluated in a transcriptional activation assay with hAR in a mammalian cell background (CV-1) as the primary in vitro assay. Rece...More data for this Ligand-Target Pair

Target InfoPDBMMDBNCI pathwayReactome pathwayKEGG
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Ligand InfoPC cidPC sidSimilars

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