Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetGlycylpeptide N-tetradecanoyltransferase(Trypanosoma brucei)
Univeristy Of Dundee

US Patent
LigandPNGBDBM184998(US9156811, DDD90147)
Affinity DataIC50:  34nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetGlycylpeptide N-tetradecanoyltransferase 1(Homo sapiens (Human))
Univeristy Of Dundee

US Patent
LigandPNGBDBM184998(US9156811, DDD90147)
Affinity DataIC50:  939nMpH: 7.4 T: 2°CAssay Description:Measurement of the ability of compounds to inhibit the NMT-1 and/or NMT-2 enzyme isoforms of human, trypanosome (T. brucei), leishmanial (L. major) a...More data for this Ligand-Target Pair
In DepthDetails US Patent