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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Adenosine receptor A1
(GUINEA PIG)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50004588
(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-isobuty...)
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Affinity Data
Ki: 15nM
Assay Description:
Binding affinity against adenosine A1 receptor in guinea pig forebrain membranes using N6-[3H]cyclohexyladenosine as radioligand
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Adenosine receptor A1
(GUINEA PIG)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50004588
(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-isobuty...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 15nM
Assay Description:
Inhibition of N6-[3H]cyclohexyladenosine binding to guinea pig forebrain membrane Adenosine A1 receptor
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A2a/A2b
(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50004588
(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-isobuty...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 850nM
Assay Description:
Binding affinity against Adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide in rat striatal membranes
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Adenosine receptor A2a/A2b
(Rattus norvegicus)
Kyowa Hakko Kogyo
Curated by
ChEMBL
Ligand
BDBM50004588
(8-(Hexahydro-2,5-methano-pentalen-3a-yl)-3-isobuty...)
Copy SMILES
Copy InChI
Affinity Data
Ki: 850nM
Assay Description:
Binding affinity against adenosine A2 receptor in rat striatal membranes using N-[3H]-ethyladenosin-5''-uronamide as radioligand in the presence of 5...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI