Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 5 hits in this display
BDBM50014255(7-Benzyl-3-isobutyl-1-methyl-3,7-dihydro-purine-2,...)
BDBM50014255(7-Benzyl-3-isobutyl-1-methyl-3,7-dihydro-purine-2,...)
Ki: 7.50E+3nMAssay Description:Antagonism of N-ethylcarboxamido adenosine-stimulated adenylate cyclase associated with stimulation of Adenosine A2 receptor of rat PC12 membranesMore data for this Ligand-Target Pair
BDBM50014255(7-Benzyl-3-isobutyl-1-methyl-3,7-dihydro-purine-2,...)
Ki: 9.00E+3nMAssay Description:Ability to inhibit binding of 1 nM [3H]-cyclohexyladenosine to adenosine A1 receptor in rat cerebral cortical membranesMore data for this Ligand-Target Pair
BDBM50014255(7-Benzyl-3-isobutyl-1-methyl-3,7-dihydro-purine-2,...)
Ki: 1.10E+4nMAssay Description:Compound was evaluated for its ability to antagonise cyclic [3H]-AMP accumulation in [3H]-adenine-labeled guinea pig cerebral cortical slices.More data for this Ligand-Target Pair
BDBM50014255(7-Benzyl-3-isobutyl-1-methyl-3,7-dihydro-purine-2,...)