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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

LigandPNGBDBM50226946(CHEMBL288398)
Affinity DataKi:  25nMAssay Description:Binding affinity against alpha-2 adrenergic receptor was determined by the displacement of [3H]clonidine from rat brain cortical membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50226946(CHEMBL288398)
Affinity DataIC50:  95nMAssay Description:Alpha-2 adrenergic receptor antagonistic activity in rat vas deferens.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed