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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
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Target
Metabotropic glutamate receptor 1
(Homo sapiens (Human))
Tsukuba Research Institute
Curated by
ChEMBL
Ligand
BDBM50301823
(5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
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Affinity Data
IC50: 5.5nM
Assay Description:
Antagonist activity at human mGluR1 receptor expressed in CHO cell membranes assessed as inhibition of L-glutamate-induced calcium mobilization by FL...
More data for this Ligand-Target Pair
Target Info
PDB
Reactome pathway
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
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In Depth
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Article
PubMed
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Target
Metabotropic glutamate receptor 5
(Homo sapiens (Human))
Tsukuba Research Institute
Curated by
ChEMBL
Ligand
BDBM50301823
(5-(1-(2-fluoropyridin-3-yl)-5-methyl-1H-1,2,3-tria...)
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Copy InChI
Affinity Data
IC50: 2.30E+3nM
Assay Description:
Antagonist activity at human mGluR5 receptor expressed in CHO cell membranes assessed as inhibition of L-glutamate-induced calcium mobilization by FL...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI