Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetBombesin receptor subtype-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340970((+/-)-4-((endo)-bicyclo[2.2.1]heptan-2-ylamino)-N-...)
Affinity DataIC50:  820nMAssay Description:Binding affinity to human BRS3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340970((+/-)-4-((endo)-bicyclo[2.2.1]heptan-2-ylamino)-N-...)
Affinity DataEC50:  98nMAssay Description:Agonist activity at mouse BRS3 by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBombesin receptor subtype-3(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50340970((+/-)-4-((endo)-bicyclo[2.2.1]heptan-2-ylamino)-N-...)
Affinity DataEC50:  940nMAssay Description:Agonist activity at human BRS3 by functional assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed