Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 3 hits in this display   

TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388959(CHEMBL2063724)
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 5(Rattus norvegicus (Rat))
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388959(CHEMBL2063724)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of [11C]-ABP688 from mGluR5 in Sprague-Dawley rat brain homogenates after 1 hr by gamma countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
National Institute Of Radiological Sciences

Curated by ChEMBL
LigandPNGBDBM50388959(CHEMBL2063724)
Affinity DataIC50: >1.00E+4nMAssay Description:Displacement of 4-[18F]fluoro-N-[4-(6-(isopropylamino)pyrimidin-4-yl)-1,3-thiazol-2-yl]-N-methylbenzamide from mGluR1 in Sprague-Dawley rat brain hom...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed