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Compile Data Set for Download or QSAR
maximum 50k data
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
4
hits in this display
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
Wyeth Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50306031
(3-(3-(3-(isopropylsulfonyl)phenoxy)phenyl)-2-methy...)
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Affinity Data
IC50: 33nM
Assay Description:
Displacement of [3H]T0901317 from human recombinant LXRalpha LBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
Wyeth Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50306031
(3-(3-(3-(isopropylsulfonyl)phenoxy)phenyl)-2-methy...)
Copy SMILES
Copy InChI
Affinity Data
IC50: 960nM
Assay Description:
Displacement of [3H]T0901317 from human recombinant LXRbeta LBD
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-beta
(Homo sapiens (Human))
Wyeth Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50306031
(3-(3-(3-(isopropylsulfonyl)phenoxy)phenyl)-2-methy...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 4.10E+3nM
Assay Description:
Agonist activity at human Gal4-LBD fused LXRbeta LBD expressed in Huh7 cells by transient transactivation assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI
Target
Oxysterols receptor LXR-alpha
(Homo sapiens (Human))
Wyeth Pharmaceuticals
Curated by
ChEMBL
Ligand
BDBM50306031
(3-(3-(3-(isopropylsulfonyl)phenoxy)phenyl)-2-methy...)
Copy SMILES
Copy InChI
Affinity Data
EC50: 700nM
Assay Description:
Agonist activity at human Gal4-LBD fused LXRalpha LBD expressed in Huh7 cells by transient transactivation assay
More data for this Ligand-Target Pair
Target Info
PDB
UniProtKB/SwissProt
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI