Compile Data Set for Download or QSAR
maximum 50k data

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetBile acid receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50258512(3-(2-chloro-4-((3-((trans)-2-(2,6-dichlorophenyl)c...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human FXR assessed as SRC1 coactivatior peptide recruitment by cell free FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50258512(3-(2-chloro-4-((3-((trans)-2-(2,6-dichlorophenyl)c...)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at human FXR assessed as SRC1 peptide interaction with receptor ligand binding domain by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed