Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 4 hits in this display   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104324(US8575186, 197 | US8575186, 198 | US8575186, 87/18...)
Affinity DataKi:  284nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM50364989(CHEMBL1950755)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]LSD from human 5-HT6 serotonin receptor by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104324(US8575186, 197 | US8575186, 198 | US8575186, 87/18...)
Affinity DataKi:  350nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Albany Molecular Research

US Patent
LigandPNGBDBM104324(US8575186, 197 | US8575186, 198 | US8575186, 87/18...)
Affinity DataKi:  365nMAssay Description:The relative affinities of the various compounds for the 5-HT6 receptor were measured in a radioligand binding assay, using a sintillation proximity ...More data for this Ligand-Target Pair
In DepthDetails US Patent