Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)
Found 23 hits in this display
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant aurora-B expressed in Sf9 cells using tetra(LRRWSLG) as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant COT expressed in Sf9 cells assessed as autophosphorylation after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant INS-R expressed in Sf9 cells using poly(A,E,K,Y)6:2:5:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant CDK2/CyclinA expressed in Sf9 cells using histone H1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: 3.50E+4nMAssay Description:Inhibition of ABCG2 (unknown origin) expressed in HEK293 cells assessed as reduction in mitoxantrone efflux after 30 mins by FACS methodMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant AKT1 expressed in Sf9 cells using GSK3(14-27) as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant ARK5 expressed in Sf9 cells assessed as autophosphorylation after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant aurora-A expressed in Sf9 cells using tetra(LRRWSLG) as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant B-RAF expressed in Sf9 cells using MEK1 KM as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant EGF-R expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant EPHB4 expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant ERBB2 expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant FAK expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant IGF1R expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant SRC expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant VEGF-R2 expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant VEGF-R3 expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant MET expressed in Sf9 cells using poly(A,E,K,Y)6:2:5:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant PDGFRbeta expressed in Sf9 cells using poly(A,E,K,Y)6:2:5:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant PLK1 expressed in Sf9 cells using casein as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant SAK expressed in Sf9 cells using p38alpha-KRKR as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant TIE2 expressed in Sf9 cells using poly(E,Y)4:1 as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair
IC50: >3.50E+4nMAssay Description:Inhibition of human recombinant CDK4/CyclinD1 expressed in Sf9 cells using RB-CTF as substrate after 80 mins by scintillation countingMore data for this Ligand-Target Pair