Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target5-hydroxytryptamine receptor 4(Homo sapiens (Human))
Angelini Santa Palomba Research Center

Curated by ChEMBL

LigandBDBM50398983(CHEMBL2179697)Copy SMILESCopy InChI

Affinity DataKi:  0.100nMAssay Description:Displacement of [3H](1-(2-(methylsulfonamido)ethyl)piperidin-4-yl)methyl 1-methyl-1H-indole-3-carboxylate from human 5HT4R expressed in HEK293 cellsMore data for this Ligand-Target Pair

Target InfoPDBReactome pathway
UniProtKB/SwissProt
antibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI

Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
Angelini Santa Palomba Research Center

Curated by ChEMBL

LigandBDBM50398983(CHEMBL2179697)Copy SMILESCopy InChI

Affinity DataKi:  100nMAssay Description:Displacement of [3H]ketanserin from human 5HT2AR expressed in CHOK1 cellsMore data for this Ligand-Target Pair

Target InfoPDBMMDBReactome pathwayKEGG
UniProtKB/SwissProt
B.MOADDrugBankantibodypediaGoogleScholar

Ligand InfoCHEMBLPC cidPC sidSimilars

In DepthDetails ArticlePubMed
Copy BDB DOI