Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50256731(2-(1-phenylethyl)-3-p-tolyl-2,3-dihydroquinazolin-...)
Affinity DataEC50:  3.00E+3nMAssay Description:Positive allosteric modulation of human mGlu4 receptor expressed in BHK cells assessed as potentiation of glutamate-induced calcium mobilization afte...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
Lundbeck Research Usa

Curated by ChEMBL
LigandPNGBDBM50256731(2-(1-phenylethyl)-3-p-tolyl-2,3-dihydroquinazolin-...)
Affinity DataEC50:  3.00E+3nMAssay Description:Activation of human mGluR4 expressed in CHO cells coexpressing Gqi5 protein assessed as potentiation of glutamate-induced responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed