Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 5 hits in this display   

TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254543(3-(dimethylamino)butyl 3-phenylpropylcarbamate | C...)
Affinity DataKi:  91nMAssay Description:Displacement of [3H]epibatidine from alpha4beta2 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254543(3-(dimethylamino)butyl 3-phenylpropylcarbamate | C...)
Affinity DataKi:  1.40E+3nMAssay Description:Displacement of [3H]epibatidine from alpha4beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254543(3-(dimethylamino)butyl 3-phenylpropylcarbamate | C...)
Affinity DataKi:  3.98E+4nMAssay Description:Displacement of [3H]epibatidine from alpha3beta4 nAChR (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254543(3-(dimethylamino)butyl 3-phenylpropylcarbamate | C...)
Affinity DataKi: >1.00E+6nMAssay Description:Displacement of [3H]MLA from alpha7 nAChR/5HT3A receptor (unknown origin) expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-3(Homo sapiens (Human))
Copenhagen University

Curated by ChEMBL
LigandPNGBDBM50254543(3-(dimethylamino)butyl 3-phenylpropylcarbamate | C...)
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at alpha3beta4 nAChR (unknown origin) expressed in HEK293 cells by FLIPR membrane potential assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed