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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 7 hits in this display   

TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021790((S,S)1-(3-Mercapto-2-methyl-propionyl)-2,3-dihydro...)
Affinity DataIC50:  2.60nMAssay Description:Inhibition of dihydrofolate reductase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021790((S,S)1-(3-Mercapto-2-methyl-propionyl)-2,3-dihydro...)
Affinity DataIC50:  2.60nMAssay Description:Ability to inhibit Angiotensin I converting enzyme was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Rattus norvegicus)
TBA

Curated by ChEMBL
LigandPNGBDBM50421824(CHEMBL75752)
Affinity DataIC50:  3.70nMAssay Description:Inhibition of rat Angiotensin I converting enzyme (ACE), using Hip-Gly-Gly as synthetic substrate.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50406945(CHEMBL611148)
Affinity DataIC50:  6nMAssay Description:Inhibitory activity against angiotensin converting enzyme (ACE)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Homo sapiens (Human))
Washington University

Curated by ChEMBL
LigandPNGBDBM50021790((S,S)1-(3-Mercapto-2-methyl-propionyl)-2,3-dihydro...)
Affinity DataIC50:  12.6nMAssay Description:Inhibition of angiotensin I converting enzyme in silicoMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021790((S,S)1-(3-Mercapto-2-methyl-propionyl)-2,3-dihydro...)
Affinity DataIC50:  23nMAssay Description:In vitro inhibition of Angiotensin I converting enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50021790((S,S)1-(3-Mercapto-2-methyl-propionyl)-2,3-dihydro...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of dihydrofolate reductase in Escherichia coliMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed