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Compile Data Set for Download or QSAR
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
(change energy unit to
kcal/mol
)
Found
2
hits in this display
Target
11-beta-hydroxysteroid dehydrogenase 1
(Mus musculus (mouse))
Chinese Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50296708
(3-{4-{2-Amino-6-[4-(3-trifluoromethyl-benzyl)-pipe...)
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Affinity Data
IC50: 1.04E+3nM
Assay Description:
Inhibition of mouse liver microsome 11betaHSD1 expressed in HEK293 cells assessed as conversion of [3H]cortisone into [3H]cortisol by scintillation p...
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
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Target
Peroxisome proliferator-activated receptor gamma
(Homo sapiens (Human))
Chinese Academy Of Sciences
Curated by
ChEMBL
Ligand
BDBM50296708
(3-{4-{2-Amino-6-[4-(3-trifluoromethyl-benzyl)-pipe...)
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Copy InChI
Affinity Data
EC50: 4.79E+3nM
Assay Description:
Agonist activity at human PPARgamma expressed in U2OS cells by luciferase transactivation assay
More data for this Ligand-Target Pair
Target Info
PDB
MMDB
NCI pathway
Reactome pathway
KEGG
UniProtKB/SwissProt
B.MOAD
DrugBank
antibodypedia
GoogleScholar
Ligand Info
CHEMBL
PC cid
PC sid
Patents
Similars
In Depth
Details
Article
PubMed
Copy BDB DOI