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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50296708(3-{4-{2-Amino-6-[4-(3-trifluoromethyl-benzyl)-pipe...)
Affinity DataIC50:  1.04E+3nMAssay Description:Inhibition of mouse liver microsome 11betaHSD1 expressed in HEK293 cells assessed as conversion of [3H]cortisone into [3H]cortisol by scintillation p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Chinese Academy Of Sciences

Curated by ChEMBL
LigandPNGBDBM50296708(3-{4-{2-Amino-6-[4-(3-trifluoromethyl-benzyl)-pipe...)
Affinity DataEC50:  4.79E+3nMAssay Description:Agonist activity at human PPARgamma expressed in U2OS cells by luciferase transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed