Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 2 hits in this display   

TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50408699(CHEMBL2110165)
Affinity DataKi:  274nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50063199((3-Benzyl-3H-[1,2,3]triazolo[4,5-d]pyrimidin-7-yl)...)
Affinity DataKi:  575nMAssay Description:Compound was tested for binding affinity at Adenosine A1 receptor in bovine brain cortical membranes using [3H]-(R)-(-)-N6-(2-phenylisopropyl)adenosi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed