Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB (change energy unit to kcal/mol)

Found 11 hits in this display   

TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384087(CHEMBL2029549)
Affinity DataIC50:  30nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384086(CHEMBL2029548)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384088(CHEMBL2029550)
Affinity DataIC50:  40nMAssay Description:Inhibition of human recombinant SSAO/VAP1 assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMembrane primary amine oxidase(Mus musculus)
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384088(CHEMBL2029550)
Affinity DataIC50:  130nMAssay Description:Inhibition of SSAO/VAP1 in mouse adipocytes measuring H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384087(CHEMBL2029549)
Affinity DataIC50:  1.61E+3nMAssay Description:Inhibition of human recombinant MAO-B assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384087(CHEMBL2029549)
Affinity DataIC50:  2.46E+3nMAssay Description:Inhibition of human DAO measuring H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384086(CHEMBL2029548)
Affinity DataIC50:  2.98E+3nMAssay Description:Inhibition of human recombinant MAO-B assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384088(CHEMBL2029550)
Affinity DataIC50:  6.43E+3nMAssay Description:Inhibition of human recombinant MAO-B assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384088(CHEMBL2029550)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant MAO-A assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384087(CHEMBL2029549)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human recombinant MAO-A assessed as H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD-amino-acid oxidase(Homo sapiens (Human))
Pharmaxis

Curated by ChEMBL
LigandPNGBDBM50384088(CHEMBL2029550)
Affinity DataIC50:  7.41E+4nMAssay Description:Inhibition of human DAO measuring H2O2 production by Resorufin/Amplex Red assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed